Webinar

High-Throughput Screening of GPCRs for Drug Discovery Applications

What is covered in this webinar:

Case studies highlighting screening and assay development of small-molecule antagonists for GPCRs
High-throughput-screening for Gq-coupled receptors using fluorescence-based detection of second messengers
High-throughput-screening hit selection and compound profiling for GPCRs

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Speakers

Edward Ainscow

Dr. Edward Ainscow
Director, Genomics Institute of the Novartis Research Foundation.

Sylvie Jezequel-Sur

Sylvie Jezequel-Sur
MS, Associate Principal Scientist, Merck & Co.

R. Jason Kirby

R. Jason Kirby
MS, Senior Associate Scientist, Sanford Burnham Prebys Medical Discovery Institute.

Abstract

GPCRs constitute the largest class of protein targets for pharmacological manipulation. However, technical challenges persist in the rapid screening of GPCR agonists and antagonists. A panel of experts will discuss advances in high-throughput screening for GPCR drug discovery.